Nitrogen mustard compounds
Medchemexpress LLC Bis(2-chloroethyl)amine-1,1,2,2-d4 hydrochloride | 352431-06-2 | 98.0% | 182.51 | C4H6D4Cl3N | 5mg
Bis(2-chloroethyl)amine-1 1 2 2-d4 (hydrochloride) is the deuterium labeled Bis(2-chloroethyl)amine-1 1 2 2 hydrochloride[1]
Chemscene ChemScene | 4,7-Dibromoisoquinoline | 250MG | CS-0139734 | 0.97 | 223671-10-1| MFCD13191776 | 286.95
ChemScene | 4,7-Dibromoisoquinoline | 250MG | CS-0139734 | 0.97 | 223671-10-1| MFCD13191776 | 286.95
Chem-Impex International, Inc. N,N-Bis(2-chloroethyl)-p-toluenesulfonamide | MFCD00018944 | 25G
N,N-Bis(2-chloroethyl)-p-toluenesulfonamide, MFCD00018944, 25G
Medchemexpress LLC ZL0580 | 2377151-10-3 | 99.4% | 532.53 | 100 MG
ZL0580, a structurally close analog of ZL0590, induces epigenetic suppression of HIV via selectively binding to BD1 domain of BRD4. It induces HIV suppression by inhibiting Tat transactivation and transcription elongation as well as by inducing repressive chromatin structure at the HIV promoter.
- Induces epigenetic suppression of HIV
- Selectively binds to BD1 domain of BRD4
- Inhibits Tat transactivation and transcription elongation
- Induces repressive chromatin structure at the HIV promoter
- Suppresses HIV in primary CD4+ T cells
- Exhibits low toxicity in cell viability assays
![Medchemexpress LLC 5-amino-N-(3-fluoro-4-methoxybenzyl)-3,4-dimethylthieno[2,3-c]pyridazine-6-carboxamide | 1451994-10-7 | 99.3% | 50 MG](https://assets.fishersci.com/TFS-Assets/CCG/product-images/5000234776.png-250.jpg)
Medchemexpress LLC 5-amino-N-(3-fluoro-4-methoxybenzyl)-3,4-dimethylthieno[2,3-c]pyridazine-6-carboxamide | 1451994-10-7 | 99.3% | 50 MG
VU0467485 (AZ13713945) is a potent, selective, orally bioavailable positive allosteric modulator of the muscarinic acetylcholine receptor M4, provided as a research reagent for receptor pharmacology and preclinical studies.
- Potent and selective M4 positive allosteric modulator.
- Orally bioavailable properties support in vivo evaluation.
- High purity suitable for pharmacological assays.
- Available in multiple pack sizes, including 50 mg.
- Commonly used for studies of M4 signaling and antipsychotic-like activity in preclinical models.
Medchemexpress LLC ML-184 50mg | 794572-10-4 | 470.63 g/mol | C25H34N4O3S | 50 MG
ML-184 is a selective GPR55 agonist research compound (CAS 794572-10-4) used to probe GPR55-mediated signaling pathways in vitro and in vivo. It activates ERK1/2 phosphorylation, promotes PKCβII translocation, and has been shown to increase neural stem cell proliferation and differentiation.
- Selective GPR55 agonist with an EC50 of about 250 nM.
- Greater than 100-fold selectivity over GPR35, CB1, and CB2.
- Induces ERK1/2 phosphorylation and PKCβII membrane translocation.
- Demonstrated activity in neural stem cell proliferation and differentiation assays.
- Provided as a high-purity solid and as a DMSO solution for biological assays.
eMolecules JW PharmLab LLC / 2-(Pentafluorosulfur)aniline / 50mg / 722712393 / 20R2505 / 96.000 / 1246998-10-6 / MFCD21362226 / 219.170 / C6H6F5NS
JW PharmLab LLC / 2-(Pentafluorosulfur)aniline / 50mg / 722712393 / 20R2505 / 96.000 / 1246998-10-6 / MFCD21362226 / 219.170 / C6H6F5NS
Medchemexpress LLC Mizagliflozin | 666843-10-3 | 99.2% | 564.67 | 5 MG
Mizagliflozin (DSP-3235 free base) is a potent, orally active, and selective SGLT1 inhibitor with a Ki of 27 nM for human SGLT1. It shows 303-fold selectivity over SGLT2. Mizagliflozin is used as an antidiabetic agent that can modify postprandial blood glucose excursion. It also exhibits potential in the amelioration of chronic constipation.
- Potent, orally active, and selective SGLT1 inhibitor (Ki of 27 nM for human SGLT1)
- 303-fold selectivity over SGLT2
- Solid appearance, off-white to light yellow color
- Used as an antidiabetic agent to modify postprandial blood glucose excursion
- Exhibits potential in the amelioration of chronic constipation
![Medchemexpress LLC 5-amino-N-[(3-fluoro-4-methoxyphenyl)methyl]-3,4-dimethylthieno[2,3-c]pyridazine-6-carboxamide | 1451994-10-7 | 99.3% | 5 MG](https://assets.fishersci.com/TFS-Assets/CCG/product-images/5000234498.png-250.jpg)
Medchemexpress LLC 5-amino-N-[(3-fluoro-4-methoxyphenyl)methyl]-3,4-dimethylthieno[2,3-c]pyridazine-6-carboxamide | 1451994-10-7 | 99.3% | 5 MG
VU0467485 is a potent, selective, and orally bioavailable positive allosteric modulator of the muscarinic acetylcholine receptor M4, supplied as a solid research compound for in vitro and in vivo pharmacology studies.
- Potent M4 positive allosteric modulator.
- High purity (99.29%).
- Molecular formula C17H17FN4O2S and molecular weight 360.41 g·mol⁻1.
- Light yellow to yellow solid appearance.
- Available in small solid quantities for research, including 5 MG packaging.
Medchemexpress LLC RV01 | 1016897-10-1 | 98.1% | 263.29 g/mol | C17H13NO2 | 10MG
RV01 is a resveratrol analogue used as a research tool to probe ALDH2-related pathways and oxidative stress. It inhibits DNA damage, reduces ethanol-induced ALDH2 mRNA expression, scavenges hydroxyl radicals, and decreases iNOS expression, indicating anti-neuroinflammatory activity. Supplied as a powder for biochemical and cell-based research applications.
- Inhibits DNA damage and reduces ALDH2 mRNA expression.
- Scavenges hydroxyl radicals, indicating antioxidant activity.
- Decreases iNOS expression and exhibits anti-neuroinflammatory effects.
- Provided as a research-grade powder suitable for biochemical studies.
- High purity for reliable experimental results.
Medchemexpress LLC Cdc25b-in-1 | 2374831-10-2 | 98.1% | 321.37 g/mol | C20H19NO3 | 10MG
CDC25B-IN-1 is a small-molecule research inhibitor of the cell division cycle 25B (CDC25B) phosphatase, referred to in the literature as compound 4a. It is provided as a 10 mg research sample (CAS 2374831-10-2) for biochemical and cellular studies targeting CDC25B-mediated signaling.
- Potent CDC25B inhibition with reported Ki of 8.5 μM.
- High purity suitable for research (≈98.1%).
- Molecular weight 321.37 g/mol; formula C20H19NO3.
- Suitable for in vitro biochemical and cell-based assays.
- Storage under nitrogen recommended; refrigerated at 4°C; in solvent: -80°C (6 months) or -20°C (1 month).
- Supplied as a small quantity research sample for laboratory use.
Medchemexpress LLC 2-phenylaminoadenosine | 53296-10-9 | MFCD00055119 | 98.0% | 358.35 g/mol | C16H18N6O4 | 5 MG
CV1808 (2-phenylaminoadenosine) is a research-grade, non-selective A2 adenosine receptor agonist used in pharmacology and receptor-binding studies. It shows reported Ki values of 76 nM at the A2A receptor and 1,450 nM at the A3 receptor, has molecular formula C16H18N6O4 and molecular weight 358.35 g/mol, and is supplied as a solid with analytical purity around 98.0% for research use only.
- Non-selective A2 adenosine receptor agonist
- Reported Ki: A2A = 76 nM; A3 = 1,450 nM
- Molecular formula C16H18N6O4; molecular weight 358.35 g/mol
- Analytical purity approximately 98.0%
- Supplied as a solid for laboratory research applications
Medchemexpress LLC Metarrestin | 1443414-10-5 | 99.9% | 50 MG
Metarrestin is a small-molecule perinucleolar compartment inhibitor provided as a high-purity research compound for in vitro and in vivo studies investigating nucleolar structure and metastasis.
- Provides high purity (99.9%).
- Molecular formula C31H30N4O and molecular weight 474.60 g/mol.
- Available in solid and solution formats for flexibility in experiments.
- Suitable for use in biochemical, cell-based, and pharmacokinetic studies.
- Recommended storage: powder at -20°C; in solvent at -80°C.
eMolecules Synthonix - Stock / NN3-Trimethylazetidin-3-amine hydrochloride / 250mg / 525923583 / T1329 / / 132771-10-9 / MFCD22123304 / 150.650 / C6H15ClN2
Synthonix - Stock / NN3-Trimethylazetidin-3-amine hydrochloride / 250mg / 525923583 / T1329 / / 132771-10-9 / MFCD22123304 / 150.650 / C6H15ClN2
eMolecules AstaTech / PYRIDINE-2356-TETRAAMINE 3HCL / 0.1g / 722706699 / C15643 / 97.000 / 34981-10-7 / MFCD00235198 / 248.540 / C5H12Cl3N5
AstaTech / PYRIDINE-2356-TETRAAMINE 3HCL / 0.1g / 722706699 / C15643 / 97.000 / 34981-10-7 / MFCD00235198 / 248.540 / C5H12Cl3N5